[26P1-pm2-001] Synthesis of fluorescence-labeled thallusin derivatives and their effects on zoospores of green alga Gayralia

○Momoka Takahashi¹, Naoto Yamasaki¹, Masaya Takehara¹, Tomoyuki Esumi¹, Hiromichi Kennmoku¹, Yoshinori Asakawa¹, Hirohumi Yamamoto¹ (1. Pharm. Sci., Tokushima bunri Univ.)

[26P1-pm2-002S] Development of N-fluoroalkylation for various nitrogen-containing heterocycles

○Yukari Akamatsu¹, Kohei Hamayasu¹, Yukiko Karuo¹, Atsushi Tarui¹, Kazuyuki Sato¹, Kentaro Kawai¹, Masaaki Omote¹ (1. Faculty of Pharmaceutical Sciences, Setsunan University)

[26P1-pm2-003S] Synthetic study of indole-pyrazole type bi-heteroaryl compounds under the common Suzuki coupling conditions

○Natsuki Honda¹, Takuya Okawauchi¹, Ryota Fujimoto¹, Noriyuki Nakajima^1,2, Yasuhito Koyama^1,2, Masahiro Hamada^1,2 (1. Toyama Prefectural University, 2. Biotech. Res. Center, Toyama Pref. Univ.)

[26P1-pm2-004] A concise synthetic route to nobiletin

○Yuka Takahashi¹, Hidetsugu Tabata¹, Tetsuta Oshitari¹ (1. Faculty of Pharma Sciences, Teikyo University)

[26P1-pm2-005S] Synthetic study of specific inhibitors toward a peptide epimerase MurL

○Takumi Yamaoka¹, Fumihiro Isikawa¹, Yasushi Ogasawara², Tohru Dairi², Genzoh Tanabe¹ (1. Faculty of Pharmacy, Kindai University, 2. Graduate School of Engineering, Hokkaido University)

[26P1-pm2-006] Synthesis of antitumor cyclic hexapeptide RA-VII analogues with an aromatic amino acid at position 2. Part II.

○Motoki Katoh¹, Keiichiro Ogura¹, Tomoyo Hasuda¹, Haruhiko Fukaya¹, Yukio Hitotsuyanagi¹ (1. Tokyo Univ. of Pharm. & Life Sci., Sch. of Pharm.)

[26P1-pm2-007S] Evaluation of H-bonding Ability of Chloroalkene Dipeptide Isosteres Using Peptide Catalyst System

○Chihiro Iio¹, Fujimoto Junko², Toyama Daichi¹, Sato Kohei^1,2, mase Nobuyuki^1,2, Narumi Tetsuo^1,2 (1. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ., 2. Fac. Eng., Shizuoka Univ.)

[26P1-pm2-008S] Synthesis of amide-to-fluoroalkene peptidomimetic of
Aβ-derived peptide containing Phe-Phe-type fluoroalkene dipeptide isostere

○Ai Sakakibara¹, Chihiro Iio², Kohei Sato^1,2, Nobuyuki Mase^1,2, Tetsuo Narumi^1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ.)

[26P1-pm2-009] Synthesis of a disaccharide, Emmyguyacins B, containing anti influenza virus.

○Isao Ohtsuka¹, Toshiyuki Atsumi¹ (1. Kyushu University Health and Welfare)

[26P1-pm2-010] Effects of sulfated vizantin based on docking simulation analysis

○Yui Asano¹, Naoto Yamasaki¹, Hironobu Takahashi¹, Tomoyuki Esumi, Kenmoku Hiromichi¹, Yoshinori Asakawa¹, Hirofumi Yamamoto¹ (1. Facalty of Pharmaceutical Science, Tokushima Bunri University)

[26P1-pm2-011S] Efforts toward Synthesis of Pericosine E Analogs Bearing A Halogen Atom Other Than Chlorine

○Keika Miyamoto¹, Saya Atarashi¹, Arisa Nomura¹, Yoshihiro Uesawa², Noboru Hayama¹, Hiroki Yoneyama¹, Yoshihide Usami¹ (1. Fac. Pharm., Osaka Med. Pharm. Univ., 2. Meiji Pharm. Univ.)

[26P1-pm2-012] Synthetic study of C-linked trehalose analogues

Rintaro Nakahashi¹, Takahiro Moriyama¹, ○Hiroaki Matoba¹, Makoto Yoritate¹, Go Hirai¹ (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)

[26P1-pm2-013] Synthesis of novel entecavir analogues having cyano group and fluorine; Evaluation of their anti-HBV activity

○HIROKI KUMAMOTO¹, Nobuyo Kuwata Higashi², Sanae Hayashi³, Debananda Das⁴, Haydar Bulut⁴, Ryoh Tokuda⁵, Shukei Imoto⁵, Kengo Onitsuka², Yuka Honda⁶, Yuki Odanaka⁶, Satoko Matsubayashi Shinnbara⁶, Kazuhiro Haraguchi¹, Yasuhito Tanaka³, Hiroaki Mitsuya^2,4 (1. Department of Pharmaceutical Sciences, Nihon Pharmaceutical University, 2. NCGM, 3. Kumamoto University, 4. NIH, 5. Sojo University, 6. Showa University)

[26P1-pm2-014S] Photoracemization of chiral sulfoxides by using photocatalysts

○Saki Fukushima¹, Kumi Tozawa¹, Kosho Makino², Kayo Nakamura¹, Hidetsugu Tabata³, Tetsuta Oshitari³, Hideaki Natsugari⁴, Hideyo Takahashi¹ (1. Pharm.Sci., Tokyo University of Science., 2. Pharm.Sci., Musashino Univ., 3. Pharm.Sci., Teikyo Univ., 4. Pharm.Sci., Tokyo Univ.)

[26P1-pm2-015S] Development of a synthesis method for various fluoroalkenes using Suzuki-Miyaura cross-coupling

○Keita Hirata¹, Yukiko Karuo¹, Atushi Tarui¹, Kazuyuki Sato¹, Kentaro Kawai¹, Masaaki Omote¹ (1. Faculty of Pharmaceutical Sciences, Setsunan University)

[26P1-pm2-016] Synthesis of optically pure erythro-2-amino-1,2-bis(4-methoxyphenyl)ethan-1-ol via Lipase TL-mediated kinetic resolution of anisoin

○Saya Okumura¹, Monami Tsukamoto¹, Yukiko Otake¹, Reiko Yano¹, Yukio Hitotsuyanagi², Yutaka Aoyagi¹, Robert M. Williams³ (1. Coll. of Pharm., Kinjo Gakuin Univ., 2. School of Pharm., Tokyo Univ. of Pharm. and Life Sci., 3. Depart. of Chem., Colorado State Univ.)

[26P1-pm2-017] Synthesis of biosynthetic intermediates of vibrioferrin and enzymatic reactions using them as substrates

○Hidemichi Mitome¹, Tomotaka Tanabe¹, Tatsuya Funahashi¹, Kazuki Akira¹ (1. Col. Pharm. Sci., Matsuyama Univ.)

[26P1-pm2-018] A synthetic method for enyne compounds using highly halogenated alkenes

○yukiko karuo¹, Atsushi Tarui¹, Kazuyuki Sato¹, Kentaro Kawai¹, Masaaki Omote¹ (1. Faculty of Pharmaceutical Sciences, Setsunan University)

[26P1-pm2-019S] Construction of successive three asymmetric carbons toward synthesis of rearranged-vibsanines

○SHINO BANDO¹, KENICHI HARADA¹, DAI HAMAMOTO¹, MIWA KUBO¹, YOSHIYASU FUKUYAMA¹ (1. Tokushima Bunri University)

[26P1-pm2-020] Synthetic studies of polymers from half-esters having the norbornadiene skeleton by ring-opening metathesis polymerizations and the saturated derivatives

Xiaoxue Lin², Jianjun Shi^1,2, ○Satomi Niwayama¹ (1. Grad. Sch. Eng., Muroran Institute of Technology, 2. Grad. Sch. Chem. Eng.,Hainan Normal University)

[26P1-pm2-021] Synthesis of 14β-estradiol to improve estrogen β receptor selectivity

Hinako Sato¹, Takayuki Kanaya¹, Noriyuki Kogure¹, ○Kohei Inomata¹ (1. Pharm. Sci., Int. Univ. Health and Welfare)

[26P1-pm2-022S] Synthetic study of sphingomyelinase inhibitor SMY-540 analogues.

○Mao Yamaguchi¹, Shino Inishi¹, Kotono Kamei¹, Yusuke Kasai¹, Hiroshi Imagawa¹ (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[26P1-pm2-023S] A short-step synthesis for optically active norbornane derivative with lactam structure

○Mayu Terauchi¹, Hiroto Kaku¹, Natsuki Kyan¹, Natsumi Tada¹, Jinuk Lee¹, Yuki Ujihara¹, Kei Kitamura¹, Tetsuto Tsunoda¹ (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[26P1-pm2-024] Development of a synthetic method for dihydrosphingomyelin and Its application for RNA delivery

○Rina Fujihara¹, Yuki Nakasaku¹, Naofumi Fukata¹, Kimitada Terao¹ (1. nippon fine chemical co., ltd.)

[26P1-pm2-025S] Asymmetric total synthesis of β-carboline alkaloid (S)-brevicolline as antiviral agents.

○Koharu Sakoguchi¹, Takashi Nishiyama¹, Ryouya Shouno¹, Natsumi Nakanishi¹, Manami Obata¹, Tominari Choshi¹ (1. Fukuyama Univ.)

[26P1-pm2-026S] Total synthesis of camptothecin analogues rosettacin and synthesis of its derivatives

○Shota Mizuno¹, Takashi Nishiyama¹, Mai Endo¹, Takaki Yoshiura¹, Toshio Motoyashiki¹, Noriyuki Hatae², Tominari Choshi¹ (1. Fukuyama Univ., 2. Yokohama univ. of pharm.)

[26P1-pm2-027S] Total synthesis indolo[3,2-a]carbazole alkaloid racemosin B

○Nanaka Fukada¹, Takashi Nishiyama¹, Yuria Takeo¹, Tominari Choshi¹ (1. Fukuyama University)

[26P1-pm2-028] Total synthesis of calothrixin B and its analogs.

○Takashi Nishiyama¹, Yushi Yamaguchi¹, Aoi Okubo¹, Haruna Okihara¹, Toshio Motoyashiki¹, Noriyuki Hatae², Tominari Choshi¹ (1. Fukuyama Univ., 2. Yokohama univ. of pharm.)

[26P1-pm2-029S] Synthesis of novel pyridoimidazoisoquinoliniums via silver-mediated intramolecular cyclization and application for live cell imaging

○Masato Kawakubo¹, Yoshikazu Inoh¹, Yuki Murata¹, Mio Matsumura¹, Tadahide Furuno¹, Shuji Yasuike¹ (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[26P1-pm2-030] Synthesis of 2-aminodibenzo[d,f][1,3]oxazepines from 2′-amino-2-hydroxybiphenyl and isothiocyanates via iodine-mediated cyclodesulfurization

○Yuki Murata¹, Arisu Koyanagi¹, Mako Izawa¹, Yukako Hayashi², Tadashi Hyodo², Mio Matsumura¹, Kentaro Yamaguchi², Shuji Yasuike¹ (1. Sch. Pharm. Sci., Aichi Gakuin Univ., 2. Sch. Phram Sci., Tokushima Bunri Univ.)

[26P1-pm2-031S] Synthesis of 2-arylbenzoazoles from thioamides and aminophenols via Ph₃BiCl₂-promoted desulfurization

○Arisu Koyanagi¹, Yuki Murata¹, Shiori Hayakawa¹, Mio Matsumura¹, Shuji Yasuike¹ (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[26P1-pm2-032] Syntehsis of 5-FU selene analog: Ag catalyzed regioselective C-H selenation of uracils

○Mio Matsumura¹, Saori Tsuchida¹, Rena Nezaki¹, Yuki Murata¹, Shuji Yasuike¹ (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[26P1-pm2-033] Synthetic Studies of Novel Heterocyclic Linking Pyrazole Derivatives based on 4-Hydroxypyrazoles

Eiichi Masumoto¹, ○Saori Shindo¹, Kohei Kobayashi¹, Fumi Okabe-Nakahara¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[26P1-pm2-034S] Synthetic Studies of Novel Spiro-1,3,4-Oxaziazole-Pyrazolone Derivatives

Eiichi Masumoto¹, ○Kazutoshi Ihara¹, Hanae Seki¹, Fumi Okabe-Nakahara¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[26P1-pm2-035] Synthetic Studies of fused tricyclic imidazo[1,2-a]pyridine derivatives.

Fumi Okabe-Nakahara¹, ○Yuuna Mihara¹, Eiichi Masumoto¹, Hiroshi Maruoka¹ (1. Fac. Pharm. Sci., Fukuoka Univ.)

[26P1-pm2-036S] Synthetic Studies of Matrine Analogues

○Hana Uemura¹, Haruki Obata¹, Takeshi Noda² (1. Kanagawa Institute of Technology, 2. Kanagawa institute of technology)

[26P1-pm2-037S] Synthetic Studies of Sparteine and Anagyrine Analogues

○Daiki Arai¹, Takeshi Noda² (1. Kanagawa Institute of Technology, 2. Kanagawa institute of technology)

[26P1-pm2-038S] Synthetic Studies of New Bicyclic Pipecolic Acid Derivatives

○Masahiko Yamamoto¹, Takeshi Noda² (1. Kanagawa Institute of Technology, 2. Kanagawa institute of technology)

[26P1-pm2-039] Synthesis and properties of 4-chloropyrimidine-C-nucleoside for inhibition of DNA cytosine-5 methyltransferase (DNMT)

○Kousuke Sato¹, Yuria Chiba¹, Mayu Ohyama¹, Takahiro Sasaki¹, Tsuyoshi Murai¹ (1. Sch. Pharm. Sci., Health Sci. Univ. Hokkaido)

[26P1-pm2-040] Design and synthesis of ApoB-targeted prodrug siRNA containing partial modifications for improvement of nuclease resistance

○Junsuke Hayashi¹, Yosuke Ochi¹, Shun-ichi Wada¹, Fumito Wada², Mariko Harada-Shiba², Hidehito Urata¹ (1. Osaka Med. and pharm. Univ., 2. National Cerebral and Cardiovascular Center)

Session information

[26P1-pm2] Total synthesis/Biosynthesis/Other synthetic studies

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