Session information

Academic Program (AP)

Chemical Biology

Chemical Biology

Mon. Mar 18, 2019 1:00 PM - 6:30 PM F6 (356, Bldg. 3 [5F])

3F6-25～3F6-29　KOWADA, Toshiyuki
3F6-32～3F6-36　SHINDO, Naoya
3F6-39～3F6-43　TAKAOKA, Yosuke
3F6-46～3F6-50　MIKI, Koji
3F6-53～3F6-57　TANAKA, Hiroshi

PM

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1:00 PM - 1:10 PM

[3F6-25] Development of a novel strain-release warhead for irreversible inhibitors.

Oral A

○TOKUNAGA, Keisuke; SHINDO, Naoya; OJIDA, Akio (Grad. Sch. Pharm., Kyushu Univ.)

PC Setting Time : 12:50 - 13:00

1:10 PM - 1:20 PM

[3F6-26] Development of third generation type EGFR covalent inhibitors using CFA chemistry

Oral A

○XIAOLIN, Guo; NAOYA, Sindo (Grad. Sch. Pharm., Kyushu Univ.)

PC Setting Time : 12:50 - 13:00

1:20 PM - 1:30 PM

[3F6-27] Toward expeditious development of photoaffinity probes by click reactions of azido-substituted aryltrifluoromethyldiazirines

Oral A

○WATANABE, Kenji; TSUDA, Junpei; OCHIAI, Hidenori; NIWA, Takashi; HOSOYA, Takamitsu (RIKEN BDR; IBB, Tokyo Med. and Dental Univ.)

PC Setting Time : 12:50 - 13:00

1:30 PM - 1:40 PM

[3F6-28] The development of a multi-functional probe which site-specifically bridges between two cysteine residues in proteins

Oral A

○HIGASHI, Sayaka; KIKUMA, Takashi; TAKEDA, Yoichi (Grad. Sch. Life Sci., Ritsumeikan Univ.)

PC Setting Time : 12:50 - 13:00

1:40 PM - 2:00 PM

[3F6-29] Selective chemical protein modification with nickel(II) and arylboronic acid

Oral B

○HANAYA, Kengo; OHATA, Jun; MILLER, Mary K.; MANGUBAT-MEDINA, Alicia E.; BALL, Zachary T. (Fac. Pharm., Keio Univ.)

PC Setting Time : 12:50 - 13:00

2:10 PM - 2:20 PM

[3F6-32] Controled enantiodifferentiating photocyclodimerization of 2-anthracenecarboxylic acid mediated by chaperonin

Oral A

○KOBAYASHI, Kota; NISHIJIMA, Masaki; ARAKI, Yasuyuki; WADA, Takehiko; KOIKE, Ayumi (Grad. Sch. Eng., KAIT; IMRAM, Tohoku Univ.)

PC Setting Time : 14:00 - 14:10

2:20 PM - 2:30 PM

[3F6-33] Development of methotrexate derivatives for reversible photo-control of binding to protein

Oral A

○MASHITA, Takato; KOWADA, Toshiyuki; TAKAHASHI, Hiroto; MATSUI, Toshitaka; MIZUKAMI, Shin (IMRAM, Tohoku Univ.)

PC Setting Time : 14:00 - 14:10

2:30 PM - 2:40 PM

[3F6-34] Design and synthesis of caged RyR antagonists with cell targeting ability

Oral A

○YOKOYAMA, Aika; FURUTA, Toshiaki (Fac. Sci., Toho Univ.)

PC Setting Time : 14:00 - 14:10

2:40 PM - 2:50 PM

[3F6-35] Photo-regulation of protein dimerization using protein labeling system

Oral A

○KOWADA, Toshiyuki; ARAI, Keisuke; YOSHIMURA, Akimasa; MATSUI, Toshitaka; KIKUCHI, Kazuya; MIZUKAMI, Shin (IMRAM, Tohoku Univ.)

PC Setting Time : 14:00 - 14:10

2:50 PM - 3:10 PM

[3F6-36] Noncovalently Caged Proteins with Molecular Glues

Oral B

○MOGAKI, Rina; OKURO, Kou; AIDA, Takuzo (Grad. Sch. Eng., The Univ. of Tokyo)

PC Setting Time : 14:00 - 14:10

3:20 PM - 3:30 PM

[3F6-39] Development of Anionic pH-Responsive Cyanine Dyes as Photoacoustic Sensors

Oral A

○MU, Huiying; TANAKA, Kouki; OE, Masahiro; MIKI, Koji; OHE, Kouichi (Grad. Sch. Eng., Kyoto Univ.)

PC Setting Time : 15:10 - 15:20

3:30 PM - 3:40 PM

[3F6-40] Synthesis of Cyanine Dyes with Fluorescence Intensity Enhanced by Formation of Cyclic Structure and Their Application as Enzyme Sensors

Oral A

○OE, Masahiro; MU, Huiying; MIKI, Koji; OHE, Kouichi (Grad. Sch. Eng., Kyoto Univ.)

PC Setting Time : 15:10 - 15:20

3:40 PM - 3:50 PM

[3F6-41] Stimuli-responsive Fluorescent Probe Based on 3,3’-Dihydroxy-2,2’-bipyridyl

Oral A

○TOKUNAGA, Daisuke; OE, Masahiro; MIKI, Koji; OHE, Kouichi (Grad. Sch. Eng., Kyoto Univ.)

PC Setting Time : 15:10 - 15:20

3:50 PM - 4:00 PM

[3F6-42] Development of Photoswitchable Inhibitors for Mitotic Kinesin CENP-E

Oral A

○MATSUO, Kazuya; MAFY, Noushaba; HIRUMA, Shota; UEHARA, Ryota; TAMAOKI, Nobuyuki (RIES, Hokkaido Univ.)

PC Setting Time : 15:10 - 15:20

4:00 PM - 4:20 PM

[3F6-43] Dynamic Photocontrol of CENP-E and Chromosome Movements During Cell Division

Oral B

○MAFY, Noushaba; MATSUO, Kazuya; HIRUMA, Shota; UEHARA, Ryota; TAMAOKI, Nobuyuki (RIES, Hokkaido Univ.)

PC Setting Time : 15:10 - 15:20

4:30 PM - 4:40 PM

[3F6-46] Development of potent acyl CoA-activating chemical catalysts through structure activity relationship studies

Oral A

○FURUTA, Masahiro; YAMATSUGU, Kenzo; XI, Siqi; AMAMOTO, Yoshifumi; LIU, Jiaan; KAWASHIMA, Shigehiro; KANAI, Motomu (Grad. Sch. Pharm., The Univ. of Tokyo)

PC Setting Time : 16:20 - 16:30

4:40 PM - 4:50 PM

[3F6-47] Synthesis of Aβ [18F] PET tracers composed of a styrylpyridine possessing a neopentyl-type labelling unit.

Oral A

○SONG, Ruichong; TAGO, Tetsuro; FUJIMAKI, Ryo; TATSUTA, Maho; TOYOHARA, Jyun; HIRANO, Kenichi; IWAI, Kumiko; ISHIBASHI, Kenji; TANAKA, Hiroshi (Sch. Mater. & Chem. Tech., Tokyo Tech.)

PC Setting Time : 16:20 - 16:30

4:50 PM - 5:00 PM

[3F6-48] Orientation preferences of hairpin pyrrole-imidazole polyamides toward the ^mCpG site

Oral A

○SATO, Shinsuke; ASAMITSU, Sefan; BANDO, Toshikazu; SUGIYAMA, Hiroshi (Fac. Sci., Kyoto Univ.)

PC Setting Time : 16:20 - 16:30

5:00 PM - 5:10 PM

[3F6-49] Synthesis and evaluation of cyclic Pyrrole-Imidazole Polyamides

Oral A

○HIROSE, Yuki; ASAMITSU, Sefan; HASHIYA, Kaori; BANDO, Toshikazu; SUGIYAMA, Hiroshi (Fac. Sci., Kyoto Univ.)

PC Setting Time : 16:20 - 16:30

5:10 PM - 5:30 PM

[3F6-50] Design and synthesis of nosyl type diazirines in photoaffinity labelling towards the elucidation of protein-ligand binding mode

Oral B

○SAAIDIN, Aimi Suhaily; MURAI, Yuta; MONDE, Kenji (Grad. Sch. Life Sci., Hokkaido Univ.)

PC Setting Time : 16:20 - 16:30

5:40 PM - 5:50 PM

[3F6-53] Discovery of novel KDM5 selective inhibitors and their effect on cancer cells

Oral A

○MIYAKE, Yuka; ITOH, Yukihiro; HATANAKA, Atsushi; SUZUMA, Yoshinori; SUZUKI, Miki; KODAMA, Hidehiko; ARAI, Yoshinobu; SUZUKI, Takayoshi (Grad. Sch. of Med. Sci., Kyoto Pref. Univ. of Med.; Nippon Pharmaceutical Chemicals Co., Ltd,)

PC Setting Time : 17:30 - 17:40

5:50 PM - 6:00 PM

[3F6-54] Synthesis and fluorescence properties of GFP dye derivatives, benzylidene imidazolinone derivatives

Oral A

○KANAMORI, Takashi; TSUZUKI, Takayuki; YUASA, Hideya (Sch. Life Sci. Tech., Tokyo Tech.)

PC Setting Time : 17:30 - 17:40

6:00 PM - 6:10 PM

[3F6-55] First Chaperonin GroEL Cluster Immobilized on Gold Nanoparticles as Functional Materials

Oral A

○SHEN, Hao; P.K, Hashim; AIDA, Takuzo (Fac. Eng., The Univ. of Tokyo)

PC Setting Time : 17:30 - 17:40

6:10 PM - 6:20 PM

[3F6-56] Syntheses of fatty acid-zerumbone conjugates and elucidation of the mechanisms for their growth inhibition of human T-cell lymphoid Jurkat cells

Oral A

○FUJIWARA, Yuko; KASHIWAZAKI, Gengo; UTAKA, Yoshimi; ITOH, Tomohiro; KITAYAMA, Takashi (Fac. Agr., Kindai Univ.)

PC Setting Time : 17:30 - 17:40

6:20 PM - 6:30 PM

[3F6-57] Development of novel chemical tools for analysis of mode of action of plant virulence factor coronatine

Oral A

○MIYAGAWA, Saki; HAYASHI, Kengo; ISHIMARU, Yasuhiro; TAKAOKA, Yousuke; UEDA, Minoru (Grad. Sch. Sci., Tohoku Univ.)

PC Setting Time : 17:30 - 17:40