Covalent inhibition of protein-protein interaction (2) : Structure-activity relationship study of covalent inhibitor based on N-acyl-N-alkyl sulfonamide (NASA) warhead

Presentation information

Academic Program (AP)

Chemical Biology

Sat. Mar 16, 2019 1:30 PM - 6:00 PM F3 (353, Bldg. 3 [5F])

1F3-28～1F3-33　MINOSHIMA, Masahumi
1F3-35～1F3-40　HAMACHI, Itaru
1F3-42～1F3-47　TSUKIJI, Shinya
1F3-49～1F3-54　TAMURA, Tomonori

2:20 PM - 2:30 PM

[1F3-33] Covalent inhibition of protein-protein interaction (2) : Structure-activity relationship study of covalent inhibitor based on N-acyl-N-alkyl sulfonamide (NASA) warhead

○SHIONO, Keiya; UEDA, Tsuyoshi; TAMURA, Tomonori; HAMACHI, Itaru (Sch. Eng., Kyoto Univ.; ERATO, JST)

PC Setting Time : 13:20 - 13:30

Keywords:covalent inhibitor、HDM2-p53 interaction、ligand-directed chemistry、in vitro

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