[28V03-pm] ヘテロ環化合物⑦

Sun. Mar 28, 2021 1:15 PM - 2:39 PM [Room V03] Oral Presentation 3 (Online)

座長：表雅章（摂南大薬）、山口英士（岐阜薬大）

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1:15 PM - 1:27 PM

[28V03-pm01] Simple synthesis of a bithiazolophane exhibiting anti-c-Met activity by acting as a hatch blocking access to the active site

○Tatsuya Takimoto¹, Hideaki Sasaki¹, Hirohito Tsue², Hiroki Takahashi², Alexander D. MacKerell³, Katsuya Nakano¹, Eori Okazaki¹, Ayumi Nakamura¹, Tatsuki Betsuyaku¹, Ryosuke Tachibana¹, Kazuhito Hioki¹, Ozge Yoluk³, Sunhwan Jo⁴ (1. Fac. Pharm. Sci., Kobe Gakuin Univ, 2. Grad. Sch. Human and Env. Studies, 3. Dept. Pharm. Sci., Sch. Pharm., Univ. of Maryland Baltimore, 4. SilcsBio, LLC)

1:27 PM - 1:39 PM

[28V03-pm02S] Elucidation of the stereoselectivity of oxime hydroxy groups by the substituent effect and application to Beckmann Rearrangement.

○Tomohiro Fujino¹, Yuko Otani¹, Tomohiko Ohwada¹ (1. Grad. Sch. Pharm. Sci., The Univ. of Tokyo)

1:39 PM - 1:51 PM

[28V03-pm03S] Synthesis and stereochemistry of triazolobenzodiazepine derivatives

○Ryoko Tanaka¹, Yuki Kanase², Kosho Makino¹, Hidetsugu Tabata², Tetsuta Oshitari², Hideaki Natsugari³, Hideyo Takahashi¹ (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma Sciences, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)

1:51 PM - 2:03 PM

[28V03-pm04S] Stereochemical property of dibenzoazepine derivatives and their biological activity

○Mayuno Hotta¹, Takuya Namba¹, Kosho Makino¹, Hidetsugu Tabata², Tetsuta Oshitari², Hideaki Natsugari³, Hideyo Takahashi¹ (1. Faculty of Pharmaceutical Science, Tokyo University of Science., 2. Faculty of Pharmaceutical Sciences, Teikyo University., 3. Faculty of Pharmaceutical Science, The University of Tokyo.)

2:03 PM - 2:15 PM

[28V03-pm05S] Asymmetric control of 1,5-benzodiazepinones based on central chirality

○Kaoru Funaki¹, Hidetsugu Tabata¹, Yusuke Nakazato¹, Yuka Takahashi¹, Tomohiko Tasaka², Hideyo Takahashi³, Hideaki Natsugari^2,4, Tetsuta Oshitari¹ (1. Faculty of Pharma Sciences, Teikyo Univerisity, 2. Affinity Science Corporation, 3. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 4. Graduate School of Pharmaceutical Sciences, The University of Tokyo)

2:15 PM - 2:27 PM

[28V03-pm06] Synthesis and characterization of dihydropyridazine-embedded aza[5]helicenes

○Kazuteru Usui¹, Ami Amano¹, Satsuki Murase¹, Tomohiro Umeno¹, Satoru Karasawa¹ (1. Faculty of Pharm. Sci., Showa Pharm. Univ.)

2:27 PM - 2:39 PM

[28V03-pm07S] Development of New Arylboronates Stable to Silica-Gel Chromatography

○Naoki Oka¹, Shuji Akai¹, Takashi Ikawa¹ (1. Grad. Sch. Pharm. Sci., Osaka Univ.)

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