[29V03-pm] 構造活性相関②

Mon. Mar 29, 2021 3:03 PM - 4:39 PM [Room V03] Oral Presentation 3 (Online)

座長：吉田将人（筑波大数理物質系）、上田篤志（長崎大院医歯薬）

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3:03 PM - 3:15 PM

[29V03-pm09S] Synthesis of Lysine Derivatives and the Application to SAR Study on Coibamide A

○Rikito Suzuki¹, Takashi Kitamura¹, Shinsuke Inuki¹, Hiroaki Ohno¹, Shinya Oishi^1,2 (1. Grad. Sch. Pharm. Sci., Kyoto Univ., 2. Dep. Med. Chem., Kyoto Pharm. Univ.)

3:15 PM - 3:27 PM

[29V03-pm10] Development of dipeptide derivative showing antibacterial activity against multidrug-resistant bacterium Stenotrophomonas maltophilia

○Koushi Hidaka^1,2, Taisei Hashimoto¹, Takumi Seki¹, Yuki Sakurai¹, Yasumitsu Sakamoto³, Saori Roppongi⁴, Mizuki Sekiya³, Akihiro Nakamura⁵, Yoshiyuki Suzuki⁶, Wataru Ogasawara⁵, Nobutada Tanaka⁷, Anna Miyazaki⁸, Keiko Hojo^1,2, Yuko Tsuda^1,2 (1. Fac. Pharm. Sci., Kobe Gakuin Univ., 2. Center Life Sci., Kobe Gakuin Univ., 3. Sch. Pharm., Iwate Med. Univ., 4. Sch. Med., Iwate Med. Univ., 5. Dept. Bioeng., Nagaoka Univ. Technol., 6. Nat. Inst. Technol., Nagaoka Col., 7. Sch. Pharm., Kitasato Univ., 8. Sch. Pharm. Pharm. Sci., Mukogawa Women's Univ.)

3:27 PM - 3:39 PM

[29V03-pm11S] A New Scaffold to Resolve the Long-standing Mystery of P2Y10’s Hydrophobic Binding Mode

○Luying Chen¹, Misa Sayama¹, Yuko Otani¹, Akiharu Uwamizu¹, Asuka Inoue², Junken Aoki¹, Tomohiko Ohwada¹ (1. Grad. Sch. Pharm. Sci., Univ. of Tokyo, 2. Grad. Sch. Pharm. Sci., Tohoku Univ.)

3:39 PM - 3:51 PM

[29V03-pm12S] Design and Synthesis of Inverse Agonists for Lipid Mediator Lysophosphatidylserine Receptors

○GE YAN¹, Misa Sayama¹, Luying Chen¹, Akiharu Uwamizu¹, Yuko Otani¹, Asuka Inoue², Junken Aoki¹, Tomohiko Ohwada¹ (1. Grad. Sch. Pharm. Sci., Univ. of Tokyo., 2. Grad. Sch. Pharm. Sci., Tohoku Univ.)

3:51 PM - 4:03 PM

[29V03-pm13S] A study on structure-activity relationship between hMATE1 and cimetidine analogues

○Susumu Shinya¹, Kentaro Kawai¹, Naoki Kobayashi¹, Yukiko Karuo¹, Atsushi Tarui¹, Kazuyuki Sato¹, Masato Otsuka¹, Masaaki Omote¹ (1. Dep. Pharm. Sci., Setsunan Univ.)

4:03 PM - 4:15 PM

[29V03-pm14] Synthesis and radical scavenging activity of novel antioxidants with nitrogen-containing substituted ortho position of 6-chromanol

○Yuta Okayama¹, Masataka Mochizuki¹, Keiko Inami¹ (1. Faculty of pharmaceutical sciences, Sanyo-Onoda City University)

4:15 PM - 4:27 PM

[29V03-pm15S] Introduction of branched structures on the cross-linking site in macrocyclic BACE1 inhibitors

○Takuya Otani¹, Kazuya Kobayashi¹, Yasunao Hattori¹, Kenichi Akaji¹ (1. Kyoto Pharm. Univ.)

4:27 PM - 4:39 PM

[29V03-pm16] Structure–activity relationship study of a promising lead compound for the development of therapeutic agent for Alzheimer's disease

○Yuki Nara¹, Tetsuya Kuga¹, Yusuke Sasano¹, Shigeki Moriguchi¹, Yoshiharu Iwabuchi¹ (1. Graduate School of Pharmaceutical Sciences, Tohoku University)

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