Poster Presentation

(A) Pharmaceutical Chemistry

[26PO7-pm1] Total synthesis-1/Other synthetic studies-1

Sat. Mar 26, 2022 1:30 PM - 3:10 PM [Room PO7] Bldgs. 3&4, 3F Passage (Bldgs. 3&4: 3F)

【説明時間】13:45～14:55

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1:30 PM - 3:10 PM

[26PO7-pm1-01S] Total Synthesis of Phenanthroviridin Aglycon

○Kohei Harasawa¹, Yuta Mori¹, Yudai Sato¹, Yusuke Akagi¹, Toshiya Komatsu¹ (1. Fac. Pharm. Sci., Teikyo Heisei Univ.)

1:30 PM - 3:10 PM

[26PO7-pm1-02S] Synthtic studies on C-mannosyl tryptophan via epoxidation of trptophanylglucal derivatives

○Tatsuya Miwa¹, Yasuhiro Nishikawa¹, Nana Okamoto¹, Tatsuaki Baba¹, Daiki Kato¹, Kazushi Yamakita¹, Natsuki Watanabe¹, Ken Ito¹, Iori Kishihata¹, Osamu Hara¹ (1. Faculty of Pharmacy, Meijo University)

1:30 PM - 3:10 PM

[26PO7-pm1-03S] Cyclotryptophyltyrosine: synthesis and crystal structure

○Ryohei Nokura¹, Haruhiko Fukaya¹, Yukio Hitotsuyanagi¹ (1. Sch. of Pharm., Tokyo Univ. of Pharm. & Life Sci.)

1:30 PM - 3:10 PM

[26PO7-pm1-04] Synthesis of antitumor cyclic hexapeptide RA-VII analogues with an aromatic amino acid at position 2

○Keiichiro Ogura¹, Motoki Kato¹, Tomoyo Hasuda¹, Haruhiko Fukaya¹, Yukio Hitotsuyanagi¹ (1. Sch. of Pharm., Tokyo Univ. of Pharm. & Life Sci.)

1:30 PM - 3:10 PM

[26PO7-pm1-05] MW-assisted Boc-based Solid-Phase Peptide Synthesis in Water

○Keiko Hojo^1,2, Suzuko Fujiwara¹, Hoshito Inai¹, Yuki Manabe¹, Yuko Tsuda^1,2 (1. Faculty of Pharmaceutical Sciences, Kobe Gakuin University, 2. Cooperative Research Center of Life, Kobe Gakuin University)

1:30 PM - 3:10 PM

[26PO7-pm1-06S] Neighboring Group Participation of Amide-to-Alkene Isosteric Switching:
Kinetic Study of the Hydrolysis Reaction of C-Terminal Esters

○Kazutoshi Kawahara¹, Sayuri Takeo², Junko Hujimoto¹, Kohei Sato^1,2, Nobuyuki Mase^1,2, Tetsuo Narumi^1,2 (1. Fac. Eng., Shizuoka., 2. Grad. Sch. Integ. Sci. Tech.)

1:30 PM - 3:10 PM

[26PO7-pm1-07S] Stereoselective Synthesis of Lys-Pro-type Fluoroalkene Dipeptide Isosteres for Probing the Effect of Prolyl Amide Bond Configurations on Tau Aggregation

○Chihiro Iio¹, Daichi Toyama², Yuki Kodama³, Kohei Sato^1,2,3, Nobuyuki Mase^1,2,3, Tetsuo Narumi^1,2,3 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ., 3. Grad. Sch. Sci. Tech., Shizuoka Univ.)

1:30 PM - 3:10 PM

[26PO7-pm1-08S] Chemical Synthesis of Hydrolysis-Resistant Ubiquitin Mimic Preventing the Formation of Multiple Bonds by Deubiquitinase

○Kohei Watanabe¹, Yoshinori Taguchi², Takuma Nishizawa², Reon Takeuchi³, Junnko Fujimoto¹, Nobuyuki Mase^1,2,3, Kohei Sato^1,2,3, Tetsuo Narumi^1,2,3 (1. Fac. Eng., Shizuoka Univ., 2. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ., 3. Grad. Sch. Sci. Tech., Shizuoka Univ.)

1:30 PM - 3:10 PM

[26PO7-pm1-09S] Identification of Peptidic Inhibitors Targeting p97-hUfd1-hNpl4 Complex

○Takaya Kawaguchi¹, Kohei Watanabe², Reon Takeuchi³, Yuki Kodama³, Mitsuo Toda^1,2, Kohei Sato^1,2,3, Nobuyuki Mase^1,2,3, Kei Okatsu⁴, Shuya Fukai⁴, Tetsuo Narumi^1,2,3 (1. Grad. Sch. Integ. Sci. Tech., Shizuoka Univ., 2. Fac. Eng., Shizuoka Univ., 3. Grad. Sch. Sci. Tech., Shizuoka Univ., 4. Grad. Sch. Sci., Kyoto Univ.)

1:30 PM - 3:10 PM

[26PO7-pm1-10S] Design and evaluation of β-cyclodextrin derivatives having multivalent carbohydrate cluster ligands for Concanavalin A

○Taro Koda¹, Hiroshi Akutsu¹, Yoshiki Oda², Takashi Yamanoi¹ (1. Fac. of. Pharm. and Pharmceut. Sci., Josai Univ., 2. Tokai university, Technology Joint Management Office)

1:30 PM - 3:10 PM

[26PO7-pm1-11S] Synthesis of a highly water-soluble β-cyclodextrin derivative and its evaluation toward sparingly soluble drugs

Taro Koda¹, ○Hayato Higuchi¹, Hiroshi Akutsu¹, Yoshiki Oda², Takashi Yamanoi¹ (1. Fac. of. Pharm. and Pharmceut. Sci., Josai Univ., 2. Tokai university, Technology Joint Management Office)

1:30 PM - 3:10 PM

[26PO7-pm1-12S] Synthesis of MGB polyamide-2'-deoxyguanosine hybrids

○Misato Takahashi¹, Aya Yamashita¹, Koichiro Ota¹, Hiroaki Miyaoka¹, Kazuo Kamaike¹ (1. Tokyo University of Pharmacy and Life Sciences )

Session information

[26PO7-pm1] Total synthesis-1/Other synthetic studies-1

[26PO7-pm1-01S] Total Synthesis of Phenanthroviridin Aglycon

[26PO7-pm1-02S] Synthtic studies on C-mannosyl tryptophan via epoxidation of trptophanylglucal derivatives

[26PO7-pm1-03S] Cyclotryptophyltyrosine: synthesis and crystal structure

[26PO7-pm1-04] Synthesis of antitumor cyclic hexapeptide RA-VII analogues with an aromatic amino acid at position 2

[26PO7-pm1-05] MW-assisted Boc-based Solid-Phase Peptide Synthesis in Water

[26PO7-pm1-06S] Neighboring Group Participation of Amide-to-Alkene Isosteric Switching:
Kinetic Study of the Hydrolysis Reaction of C-Terminal Esters

[26PO7-pm1-07S] Stereoselective Synthesis of Lys-Pro-type Fluoroalkene Dipeptide Isosteres for Probing the Effect of Prolyl Amide Bond Configurations on Tau Aggregation

[26PO7-pm1-08S] Chemical Synthesis of Hydrolysis-Resistant Ubiquitin Mimic Preventing the Formation of Multiple Bonds by Deubiquitinase

[26PO7-pm1-09S] Identification of Peptidic Inhibitors Targeting p97-hUfd1-hNpl4 Complex

[26PO7-pm1-10S] Design and evaluation of β-cyclodextrin derivatives having multivalent carbohydrate cluster ligands for Concanavalin A

[26PO7-pm1-11S] Synthesis of a highly water-soluble β-cyclodextrin derivative and its evaluation toward sparingly soluble drugs

[26PO7-pm1-12S] Synthesis of MGB polyamide-2'-deoxyguanosine hybrids

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