The 102nd CSJ Annual Meeting

Presentation information

Academic Program [Oral A]

17. Biofunctional Chemistry, Biotechnology » Oral A

[G201-4pm] 17. Biofunctional Chemistry, Biotechnology

Sat. Mar 26, 2022 1:00 PM - 3:40 PM G201 (Online Meeting)

Chair: Chiasa Uragami, Shinobu Sato

1:50 PM - 2:00 PM

[G201-4pm-06] Development of covalent inhibitors for BTK (C481S mutant) using NASA-type warhead

Shunsuke Murakawa1, Masaharu Kawano2, Tomonori Tamura2, Itaru Hamachi2,3 (1. Kyoto University, 2. Graduate school of engineering, Kyoto University, 3. JST ERATO)

[Lang.] Japanese

Keywords:covalent inhibitor, BTK, NASA, N-acyl-N-alkylsulfonamide, C481S