[28E5-pm] Structure-activity relationship

Tue. Mar 28, 2023 2:00 PM - 3:00 PM [Room E5] Institute for the Advancement of Higher Education: E201 (Bldg. E: 2F)

Chair: Yukihiro Itoh, Shinsuke Inuki

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2:00 PM - 2:12 PM

[28E5-pm01S] Synthesis of CYM51010 analoges to develop μ-δ opioid receptor heterodimer selective agonists

○Shuma Yamada¹, Haruka Yoshida^2,3, Miki Nonaka³, Kanako Miyano³, Fumika Karaki^1,2, Shigeto Hirayama^1,2, Kennosuke Itoh^1,2, Yasuhito Uezono³, Hideaki Fujii^1,2 (1. Grad. Sch. Pharm., Kitasato Univ., 2. Sch. Pharm., Kitasato Univ., 3. Dept. Pain Control Res., Jikei Univ. Sch. Med.)

2:12 PM - 2:24 PM

[28E5-pm02S] Development of the Allosteric Ligands for the Ghrelin Receptor

○Kei Ishii¹, Fumika Karaki¹, Kanako Miyano², Yasuhito Uezono², Hideaki Fujii¹ (1. Grad. Sch. Pharm. Sci., Kitasato University, 2. Dept. Pain Control Res., Jikei Univ. Sch. Med.)

2:24 PM - 2:36 PM

[28E5-pm03S] Structure-Activity Relationship Study of marinopyrrole A derivatives for Orexin Receptors

○Arisa Shinkai^1,2, Tomoya Sugai², Yukiko Ishikawa², Masashi Yanagisawa², Noriki Kutsumura^1,2 (1. College of Chemistry, University of Tsukuba., 2. IIIS, University of Tsukuba.)

2:36 PM - 2:48 PM

[28E5-pm04S] Discovery of a novel kappa opioid receptor agonist with hetero bicyclo[2.2.2]octane skeleton

○Keita Kajino^1,2, Masahiro Yata^1,2, Yasuyuki Nagumo², Akihisa Tokuda^2,3, Noriki Kutsumura^1,2,3, Tsuyoshi Saitoh^2,3, Hiroshi Nagase^1,2 (1. Deg. Prog. Pure. Appl. Sci., Univ. Tsukuba, 2. IIIS., Univ. Tsukuba, 3. Grad. Sch. Comp. Hum. Sci., Univ. Tsukuba)

2:48 PM - 3:00 PM

[28E5-pm05] Investigation of the antimicrobial activity and cytotoxicity of N-terminal (Trp-Pro-Arg)n extended derivatives of antimicrobial peptide myticalin A6 (3-23)-OH

○Keiko Okimura¹, Tatsuo Takahashi¹, Michiyo Morimoto¹, Ayaka Yamamoto¹, Tohru Daikoku¹ (1. Hokuriku University)

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