The 101st CSJ Annual Meeting

Presentation information

Academic Program [Oral A]

17. Biofunctional Chemistry, Biotechnology » Oral A

[A24-3am] 17. Biofunctional Chemistry, Biotechnology

Sun. Mar 21, 2021 9:00 AM - 11:10 AM Room 24 (Online Meeting)

Chair:Shin Mizukami, Mako Kamiya

10:00 AM - 10:10 AM

[A24-3am-07] NASA-type irreversible inhibitor for HDM2-p53 protein-protein interaction (3): Evaluation of p53 activation and cell toxicity

Itaru Hamachi1, Tomonori Tamura1, Masaharu Kawano1, Tsuyoshi Ueda1, Keiya Shiono1, Fruzsina Hobor2, Andrew Wilson2 (1. Kyoto University, 2. University of Leeds)

[Lang.] Japanese

Keywords:Irreversible inhibitor, NASA, Covalent inhibitor