The 101st CSJ Annual Meeting

Presentation information

Academic Program [Oral A]

17. Biofunctional Chemistry, Biotechnology » Oral A

[A23-4am] 17. Biofunctional Chemistry, Biotechnology

Mon. Mar 22, 2021 9:00 AM - 11:40 AM Room 23 (Online Meeting)

Chair:Tomohiro Doura, Kazuma Amaike

10:20 AM - 10:30 AM

[A23-4am-09] Rational design and functional evaluation of piperizine-based bivalent inhibitors for lipid modification of KRas

Naomi Horiuchi1, Fumitoshi Sugino1, Junko Ohkanda1 (1. Academic Assembly, Institute of Agriculture, Shinshu University)

[Lang.] Japanese

Keywords:KRas, Posttranslational lipid modification, Protein-protein interactions, Dual inhibitors, Mid-sized molecules