[29P-am001S] Development of a new drug candidate for treatment of Menkes disease

○junna tamura¹, Misaki Nakano¹, Yoshino Takahashi¹, Kayo Nakamura¹, Hidetsugu Tabata², Tetsuta Oshitari², Hideaki Natsugari³, Kosho Makino⁴, Kiyomi Ito⁴, Hideyo Takahashi¹ (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma-Science, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo, 4. Faculty of Pharmacy, Musashino University)

[29P-am002] Simple method for benzothiadiazine dioxide compounds using the redox properties of iron powder

○kyosuke kaneda^1,2, Hirotoshi Kabasawa¹, Syun Nabeki¹, Uki Matsui¹, Hiroki Sugiyama¹, Takehiro Yamagishi^1,2 (1. Pharm. Sci., HUS., 2. CRILS)

[29P-am003] Concise Synthesis of Dehydroanthophyine Derivative with Antimalarial Activity

○Hibiki Tomimori¹, Naoto Yamasaki¹, Yoshinori Asakawa¹, Hirofumi Yamamoto¹ (1. Faculy of Pharmaceutical Sciences Tokushima Bunri University)

[29P-am004S] Synthetic studies on tricyclic compounds using 1,3-dipolar cycloaddition reaction

○Nanako Oue¹, Kohei Yoshinaga¹, Satoshi Yokoshima¹ (1. Grad. Sch. Pharm. Sci., Nagoya Univ.)

[29P-am005] Side-chain fluorination of 25-hydroxyvitamin D₃ and their biological activity

○Fumihiro Kawagoe¹, Sayuri Mototani¹, Kaori Yasuda², Hiroki Mano², Toshiyuki Sakaki², Atsushi Kittaka¹ (1. Faculty Pharm. Sci., Teikyo Univ., 2. Faculty of Engineering, Toyama Prefectural Univ.)

[29P-am006S] Synthesis and crystal structure analysis of a series of Ac₃c peptides having a sulfonamide group at N-terminus

○Kazuma Kondo¹, Tomokatsu Enda¹, Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am007] Seven Polymorphs of Quinoline Sulfonamides

○Shoko Kikkawa¹, Hiroki Daitoku¹, Akihiro Hirata¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am008S] Synthesis and crystal structures of Aib peptides with mesitylene- and naphthalene-sulfonamide.

○Yusuke Saiki¹, Tomoka Ishikawa¹, Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci.Toho Univ.)

[29P-am009S] Design and synthesis of electrophilic aminating reagents based on thianthrene scaffold

○Ryutaro Tawara¹, Shohei Hamada¹, Takumi Furuta¹, Yusuke Kobayashi¹ (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-am010S] Transformation of alkene with hypervalent pnictogen compound

○Nagisa Ishida¹, Yuuki Nishida¹, Shohei Hamada¹, Takumi Furuta¹, Yusuke Kobayashi¹ (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-am011S] Development of odorless dithiophosphoric acid equivalent for hydrothiolysis of nitriles

○Sakura Tsujikawa¹, Mei Ikeda¹, Shohei Hamada¹, Takumi Furuta¹, Yusuke Kobayashi¹ (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-am012S] Structure and Property of Conformationally Controlled Urea and Thiourea by Chalcogen-bonding interaction

○Yui Amijima¹, Takumi Inoue¹, Moe Ota¹, Nami Morita¹, Shohei Hamada¹, Seikou Nakamura¹, Yusuke Kobayashi¹, Takumi Furuta¹ (1. Kyoto Pharmaceutical Univ.)

[29P-am013S] Synthesis of benzodichalcogenophene structures containing selenium atom for rhodium paddlewheel complexes.

○Yuumi Ushio¹, Shohei Hamada¹, Yuusuke Kobayashi¹, Takumi Furuta¹ (1. Fac.Pharm, Kyoto Pharmaceutical University)

[29P-am014S] Synthesis of C₂-symmetrical oxoazahelicenes

○Yuki Arai¹, Ryo Ikeda¹, Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ.,)

[29P-am015S] Synthesis of azahelicenes using stereochemistry of aromatic amide and Yamamoto coupling reaction.

○Ryo Ikeda¹, Arai Yuki¹, Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am016S] Towards a synthesis of azananobelt analogs by ring fusion of cyclic aromatic amides

○Akane Ikoshi¹, Ayaka Sugiyama¹, Akito Miyakoshi¹, Hidemasa Hikawa¹, Shoko Kikkawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am017S] Synthesis of oxoazacoronenes by Yamamoto coupling using Ni(0) reagent

○Yudai Takizawa¹, Mariko Ninomiya¹, Akihiro Yokoyama², Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ., 2. Fac. Sci. Tech. Seikei Univ.)

[29P-am018S] One-step synthesis and crystal structures of spherical amides with C₃-symmetry

○Haruka Uno¹, Daiki Koike¹, Hyuma Masu², Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ., 2. CAI, Chiba Univ.)

[29P-am019S] Synthesis of novel π-conjugated hydrocarbons using McMurry coupling reaction

○Masayoshi Okazaki¹, Yuki Saito¹, Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am020S] Synthesis of tetraphenyladamantane derivatives which have fluorescent emitting moieties at the ends of their side chains

○Yurika Yoshida¹, Sae Maeda¹, Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-am021S] Synthesis and conformational chirality of macrocyclic aromatic amides having diphenyldianthracene moieties

○Hisato Takahashi¹, Taku Nakayama¹, Shoko Kikkawa¹, Hidemasa Hikawa¹, Isao Azumaya¹ (1. Fac. Pharm. Sci., Toho Univ.)

[29P-am022S] Conformational Control of Macrocyclic Peptides Utilizing Stereoisomerism of Benzamide

○Taichi Akahane¹, Akira Katsuyama¹, Satoshi Ichikawa¹ (1. Faculty of Pharmaceutical Sciences, Hokkaido Univ.)

[29P-am023S] Atropisomeric properties of thioamides

○Ryota Takano¹, Ryoko Tanaka¹, Kayo Nakamura¹, Hidetsugu Tabata², Tetsuta Oshitari², Hideaki Natsugari³, Hideyo Takahashi¹ (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharma-Science, Teikyo University, 3. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[29P-am024S] The aggregation-induced intramolecular charge-transfer luminescence of o-carbaboranyl anisole derivatives

○Yui Asano¹, Junna Ino¹, Naoto Yamasaki¹, Yoshinori Asakawa¹, Hirofumi Yamamoto¹ (1. Faculty of Pharmaceutical Sciences Tokushima Bunri University)

[29P-am025S] Steric properties and conformational preferences of N-(2-azulenyl) aromatic amides

○Mayuko Tomita¹, Ai Ito¹, Masayuki Yunoki¹, Ai Tsuchida¹, Mayuko Watanabe¹, Ayako Ishii¹, Takamasa Amaki¹, Ryu Yamasaki¹, Iwao Okamoto¹ (1. Showa Pharmaceutical University)

[29P-am026S] Development of fluorescein based near-infrared photoredox catalyst

○Masaya Oyama¹, Masaru Tanioka¹, Yuji Matsuya¹ (1. Faculty of Pharm. Sci., University of Toyama)

[29P-am027S] Peptide Design to Control Gel-to-Sol Transition Rate

○Yoshika Hara¹, Atsuya Yaguchi¹, Hirotsugu Hiramatsu², Takahiro Muraoka^1,3 (1. Grad. Sch. Eng., Tokyo Univ. of Agri. and Tech., 2. NYCU, 3. KISTEC)

[29P-am028S] Conformational behavior of N,N'-diaryl sudstituted Tf₂C=C(NR₂)₂ type push-pull ethylene

Hikaru Yanai¹, ○Masahi Shiozawa¹, Tomoki Sakaguchi¹, Takashi Matsumoto¹ (1. Tokyo Univ. Pharm. Life Sci)

[29P-am029] Evaluation of the stability of helical structure by metal ion-mediated side chain cross-linking of peptides containing picoryl esters in the side chain

○takuma kato¹, Yukino Yamamoto¹, Naoki Kosukegawa¹, Akari Yoshikawa¹, Akiko Asano¹, Mitsunobu Doi¹ (1. Osaka. Med. Pharm. Univ.)

[29P-am030S] Synthesis of peptides with amino acids protected by a photoremovable group and their conformational analyses.

○Motoki Naka¹, Tomohiro Umeno¹, Hiroyasu Takemoto¹, Atsushi Ueda², Masakazu Tanaka², Makoto Oba¹ (1. Grad. Sch. Med. Sci., Kyoto Prefecture Univ. of Medicine, 2. Grad. Sch. Biomed. Sci., Nagasaki Univ.)

[29P-am031S] Synthesis of thioamides structurally controlled by sulfur-sulfur chalcogen bonds and their application to heterocyclic compounds

○Rika Sakai¹, Takumi Inoue¹, Shohei Hamada¹, Yusuke Kobayashi¹, Takumi Furuta¹ (1. Fac. Pharm, Kyoto Pharmaceutical University)

[29P-am032] Elucidation of thermal behavior and single crystal structure determination of acetaminophen form III

○Kasumi Kihara¹, Taiji Yamamoto¹, Yasuaki Masuda¹, Hiroyasu Sato¹, Akito Sasaki¹ (1. Rigaku Corporation)

[29P-am033] Synthesis, Characterization, and DNA cleavage activity of Zn^II–Ant-[12]aneN3

○Yoshimi Ichimaru¹, Koichi Kato¹, Hiromasa Kurosaki², Masaaki Kurihara¹ (1. Fac. Pharm. Sci., Shonan Univ. Med. Sci., 2. Coll. Pharm., Kinjo Gakuin Univ.)

[29P-am034S] Synthesis of unnatural fluorinated dipeptides with protease inhibitory activity and their effects on the stereochemistry

○Airi Ginyama¹, Yuya Miyasato¹, Atsushi Tarui¹, Ryuji Yamazawa¹, Yukiko Karuo¹, Kazuyuki Sato¹, Kentaro Kawai¹, Masaaki Omote¹ (1. Pharm. Sci., Setsunan Univ.)

[29P-am035S] Synthesis and Properties of the Optically Active Ladder Oligonaphthalenes

○Misa Sakura¹, Shunsuke Noda², Takahiro Kimoto³, Keita Okada³, Yoshitane Imai³, Ayumi Imayoshi², Kazunori Tsubaki² (1. Faculty of Life and Environmental Sciences, Kyoto Prefectual University, 2. Graduate School of Life and Environmental Sciences, Kyoto Prefectual University, 3. Graduate School of Engineering, Kindai University )

[29P-am036] Development of influenza virus NA specific fluorescent probe

○Tadamune Otsubo¹, Daiki Syuto¹, Yutaka Narimichi², Tadanobu Takahashi², Yuuki Kurebayashi², Akira Minami², Fumiteru Teraoka¹, Hideyuki Takeuchi², Kiyoshi Ikeda¹ (1. Faculty of Pharm. Sci., Hiroshima International Univ., 2. Sch. Pharm. Sci., University of Shizuoka)

[29P-am037] Synthetic research on sulfate monosaccharide type anti-dengue virus drug (4)

○fumiteru teraoka¹, Takuma Miyamoto¹, Chie Ustubo², Kazuya IRJ Hirari³, Tadamune Otsubo¹, Kiyoshi Ikeda¹ (1. Grad. Sch. Pharm. Sci., Hiroshima Int. Univ., 2. Grad. Sch. Health. Sci., Kobe Univ., 3. Dpt. Food, Nutrition Scie., Aizu Jun. Univ.)

[29P-am038S] Steric Effects in Functional Amine Compounds for CO₂ Absorbent

○Hisayo Oka¹, Chika Suefusa¹, Ryo Murakami¹, Fuyuhiko Inagaki¹ (1. Fac. Pharm. Sci., Kobegakuin Univ.)

[29P-am039S] Electronic Effects in Functional Amine Compounds for CO₂ Absorption/Desorption Performance

○Sako Yoshida¹, Chika Suefusa¹, Ryo Murakami¹, Fuyuhiko Inagaki¹ (1. Fac. Pharm. Sci., Kobegakuin Univ.)

[29P-am040S] Synthesis and properties of an activator with a ahydrophobic unit for oligonucleotide synthesis

○Koichi Mizuno¹, Yuta Ito¹, Yasufumi Fuchi¹, Yoshiyuki Hari¹ (1. Fac. Pharm. Sci., Tokushima Bunri Univ.)

[29P-am041S] Development of novel bifunctional asymmetric organocatalysts

○Souki Sakai¹, Teruyuki Ota¹, Shinya Kimura¹, Masamichi Yamanaka¹, Masashi Yokoya¹ (1. Meiji Pharm. Univ.)

[29P-am042] Evaluation of temperature-responsive self-assembly behavior of 4-aminoquinoline amphiphile: Selective construction of perforated vesicles and nanofibers

○Yosuke Hisamatsu¹, Go Toriyama¹, Katsuhiro Yamamoto², Naoki Umezawa¹ (1. Grad. Sch. Pharm. Sci., Nagoya City Univ., 2. Grad. Sch. Eng., Nagoya Inst. Tech.)

[29P-am043] Efficient fluorination on vitamin D₃ side-chain using electrophilic fluorination reagent

○sayuri mototani¹, Fumihiro Kawagoe ¹, Kaori Yasuda², Hiroki Mano², Toshiyuki Sakaki², Atsushi Kittaka¹ (1. Faculty Pharm. Sci., Teikyo University, 2. Faculty of Engineering, Toyama Prefectural University)

[29P-am044] Synthesis and properties of 2-amino-4-fluoro-3-formylpyridine-C-nucleoside for covalent inhibition of protein function

○Kousuke Sato¹, Masaru Morikawa¹, Momoko Tsuruya¹, Tetsushi Yamamoto¹, Takahiro Sasaki¹, Tsuyoshi Murai¹ (1. Sch. Pharm. Sci., Health Sci. Univ. Hokkaido)

[29P-am045S] Dynamic Kinetic Resolution of 2-Phenylpropionic Acid esters by Chiral Quaternary Ammonium Salts

○Kokoro Kimura², Kawasaki Midori¹, Yatsuzuka Kenji², Shirai Ryuichi¹ (1. Grad. Sch. Pharm. Sci.,Doshisha Women's Col., 2. Fac. Pharm. Sci.,Doshisha Women's Col.)

[29P-am046S] Synthesis and evaluation of Perylene Diimides basedCO₂ absorbents

○Sayaka Kono¹, Rie Shinohara¹, Ryo Murakami¹, Fuyuhiko Inagaki¹ (1. Fac. Pharm. Sci., Kobegakuin Univ.)

[29P-am047S] Synthesis and characterization of Sulfinic acid-responsive fluorescent molecules

○Aoi Otsuki¹, Shogo Kyogaku¹, Hiroki Tanimoto¹, Takenori Tomohiro¹ (1. Dep. Pharm. Sci., Univ. Toyama)

Session information

[29P-am] Other synthetic studies 1/Structure and physical property 1/Others

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