[29P-pm001S] Synthetic approach to kainoids via α-sp³C-H cyanation of amines under red-light irradiation

○naoaki yoshihara¹, Takehiko Yoshimitsu¹ (1. Grad. Sch. Pharm. Sci., Okayama Univ.)

[29P-pm002] Aldol-type macrocyclization reaction catalyzed by peptide foldamer catalysis

○Tomohiro Umeno¹, Yuto Yamaberi², Atsushi Ueda², Makoto Oba¹, Masakazu Tanaka² (1. Grad. Sch. Med. Sci., Kyoto Prefectural Univ. of Medicine, 2. Grad. Sch. Biomed. Sci., Nagasaki Univ.)

[29P-pm003] Regio- and stereo-selective deuterium-labeling of amino acids under flow conditions

○Tsuyoshi Yamada¹, Shuta Ichihara¹, Kwihwan Kobayashi¹, Takashi Ikawa¹, Hironao Sajiki¹ (1. Gifu Pharm. Univ.)

[29P-pm004S] Asymmetric Alkylation via Remote Asymmetric Induction: A Practical Approach to the Stereoselective Synthesis of Xaa-Asp-type Chloroalkene Dipeptide Isosteres

○Mio Takeda¹, Chihiro Iio², Daichi Toyama², Kohei Sato^1,2, Nobuyuki Mase^1,2, Tetsuo Narumi^1,2 (1. Fac. Eng., Shizuoka Univ., 2. Grag. Sch. Integ. Sci. Tech., Shizuoka Univ.)

[29P-pm005] Asymmetric aza-Henry reactions using peptide-catalysts with N-terminal benzothiadiazine

○Kazuki Satou¹, Atsushi Ueda¹, Masakazu Tanaka¹ (1. Grad. Sch. Biomed. Sci., Nagasaki Univ.)

[29P-pm006S] Synthesis of tricyclic amine bearing contiguous tetrasubstituted carbons using a cyclization–3-aza-Cope–Mannich cascade

Mika Sugiyama¹, ○Kaito Tozuka¹, Yuji Mori¹, Takeo Sakai¹ (1. Fac.Pharm. Meijo Univ.)

[29P-pm007S] Photosensitizer-mediated racemization of chiral amino acid derivatives

○Ryusei Takada¹, Riku Matsuda¹, Kayo Nakamura¹, Kosho Makino², Hidetsugu Tabata³, Tetsuta Oshitari³, Hideaki Natsugari⁴, Hideyo Takahashi¹ (1. Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2. Faculty of Pharmacy, Musashino University, Faculty of Pharma-Science, 3. Faculty of Pharma-Science, Teikyo University, 4. Faculty of Pharmaceutical Sciences, The University of Tokyo)

[29P-pm008] Intramolucular Hydrophosphimylation of 2-Alkynylaryl-H-phosphinates

○Shino Nakajima¹, Kengo Ayabe¹, Ryoji Nozawa¹, Shintaro Kamio¹, Kyosuke Kaneda^1,2, Takehiro Yamagishi^1,2 (1. Department of Med. Chem., Hokkaido Univ. of Sci., 2. Creation Research Institute of Life Science in KITA-no-DAICHI, Hokkaido Univ. of Sci.)

[29P-pm009] Synthesis of π-conjugated molecules bearing P atom and their photophysical properties

○Yoshitaka Yamashita¹, Fumiya Natori¹, Shintaro Kamio¹, Kyosuke Kaneda^1,2, Takehiro Yamagishi^1,2 (1. Department of Med. Chem., Hokkaido Univ. of Sci., 2. Creation Research Institute of Life Science in KITA-no-DAICHI, Hokkaido Univ. of Sci.)

[29P-pm010S] Investigation of Desulfurative Borylation in Aqueous Solvents

○Kazuhiro Yamashita¹, Yui Hiranaka¹, Minjae Kim ¹, Hayato Sasamoto¹, Daiki Fukue¹, Taishi Ichinose¹, Manaka Maeda¹, Honami Matsumoto¹, You Nonaka¹, Kohei Yamada¹, Yasuchika Yamaguchi¹ (1. Nagasaki international university)

[29P-pm011] Development of reductive Heck arylation of unactivated olefin under mild condition

○Takahiro Shirai¹, Yusuke Migitera², Ryo Nakajima¹, Takuya Kumamoto¹ (1. Grad. Sch. Biomed. Health Sci., Hiroshima Univ., 2. Sch. Pharm. Sci., Hiroshima Univ. )

[29P-pm012] Steric Effect of Substitution on the Nitrogen in Ring-Closing Metathesis of Ene-Ynamides

○Hideaki Wakamatsu¹, Saya Matsuzaka¹, Ryoka Okamoto¹, Yuichi Yoshimura¹ (1. Fac. Pharm. Sci., Tohoku Med. Pharm. Univ.)

[29P-pm013S] Regio- and enantioselective synthesis of succinimides bearing all-carbon quaternary centers using a chiral phenanthroline-Pd catalyst

○Midori Adachi¹, Masafumi Tamura¹ (1. Dept. Pharm. Sci., Sanyo-Onoda City Univ.)

[29P-pm014S] Asymmetric Henry Reaction Using Bisoxazoline Ligands Bearing Two Fluorous Tags

Kazuki Ishihara¹, ○Toya Natsume¹, Yamato Kato¹, Narisa Takeuchi¹, Yuka Hayashi¹, Yuna Hagiwara¹, Shota Shibuya¹, Takayuki Shioiri¹, Masato Matsugi¹ (1. Grad. Sch. Agri., Meijo Univ.)

[29P-pm015S] Dehydration of tertiary alcohols under the neutral conditions using Ru/C

○Shuki Oyama¹, Shuji Akai², Yoshinari Sawama² (1. Sch. Pharm. Sci., Osaka Univ., 2. Grad. Sch. Pharm. Sci., Osaka Univ.)

[29P-pm016S] Synthesis of Acylglycosides Using Hypervalent Iodine Reagents and Their Use as Glycosyl Donors

○KANA YANASE¹, KOJI MORIMOTO^1,2, TETSUYA KAJIMOTO¹, KITA YASUYUKI² (1. Grad. Sch. Pharm. Sci., Ritsumeikan Univ., 2. Res. Org. Sci and Tech., Ritsumeikan Univ.)

[29P-pm017] Fluorous Lewis acid-catalyzed Ring-opening Reactions of 1,6-Anhydroglucopyranose

○Akihiro Yoshida¹, Miki Namiki¹, Ryo Sagara¹, Chikako Takahashi¹, Hiroshi Akutsu¹, Takashi Yamanoi¹ (1. Faculty of Pharmacy and Pharmaceutical Sciences, Josai University )

[29P-pm018] Asymmetric synthesis of benzyl alcohol using optically active 2-(tolylsulfinyl)phenyl ketones

○Toshinori Nakakita¹, Karin Shigematsu², Yoshinori Okuno¹, Yasuo Sato¹, Masashi Asai¹, Yasuhito Nobushi², Masaharu Toriyama², Motofumi Miura² (1. YOKOHAMA UNIVERSITY OF PHARMACY, 2. SCHOOL OF PHARMACY. NIHON UNIVERSITY)

[29P-pm019S] Development of the butenolide radical-mediated dimerization

○Mizuki Oda¹, Maho Naito¹, Souhei Teshigawara¹, Tohru Nagamitsu¹, Masaki Ohtawa¹ (1. Sch. Pharm., Kitasato Univ.)

[29P-pm020] Effects of Reactant 1,3-Cyclohexanedione on Catalytic Reactions: Limiting the Loading Enables the Use of Less Catalyst in Spiro Ring Formations

○Muhammad Sohail¹, Fujie Tanaka¹ (1. Okinawa Institute of Science and Technology Graduate University)

[29P-pm021S] Synthesis of cyclic acetal by MHAT/RPC mechanism

○Takuma Sugimura¹, Bartłomiej Szarłan², Hiroki Shigehisa¹ (1. Musashino Univ., 2. Adam Mickiewicz Univ.)

[29P-pm022] Alkynyl thioesters in halocyclization/oxidative aromatization to form thiophenes

Miari Kurihara¹, Airi Ide¹, ○hiroki shigehisa¹ (1. Musashino Univ.)

[29P-pm023] Electrophilic epoxidation of α,β-unsaturated oximes and following ring-opening

○Yoshimitsu Hashimoto¹, Kiwamu Yoshida¹, Miyu Furugoori¹, Toru Yoshino¹, Kosaku Tanaka III¹, Nobuyoshi Morita¹, Osamu Tamura¹ (1. Showa Pharm. Univ.)

[29P-pm024S] Catalytic Enantioselective Mannich Reactions of Ketones with Cyclic Ketimino Esters and Their Reverse Retro-Mannich Reactions to Afford Tetrasubstituted α-Amino Acid Derivatives

○Kuan-Lin Chen¹, Fujie Tanaka¹ (1. Okinawa Institute of Science and Technology Graduate University)

[29P-pm025S] Three-component coupling reaction by direct generation of nitrones and its application

○Ayaka Yamamoto¹, Tatsuya Kouchi¹, Riku Saito¹, Kosaku Tanaka,Ⅲ¹, Yoshimitsu Hashimoto¹, Nobuyoshi Morita¹, Osamu Tamura¹ (1. Showa Pharm. Univ.)

[29P-pm026] DMAPO/Boc₂O-Mediated One-Pot Direct N-Acylation of Less Nucleophilic N-Heterocycles with Carboxylic Acids

○atsushi umehara¹, Soma Shimizu¹, Makoto Sasaki¹ (1. Grad. Sch. Life Sci. Tohoku Univ.)

[29P-pm027S] Palladium on carbon-catalyzed conversion of azides to nitriles

○Takanori Kitazono¹, Naoya Sakurada¹, Seiya Ohtori¹, Takashi Ikawa¹, Tsuyoshi Yamada¹, Hironao Sajiki¹ (1. Gifu Pharm. Univ.)

[29P-pm028] Synthesis of sulfonium salts from arylbenziodoxaborole with sulfides

○Akira Yoshimura¹, Mekhman s Yusubov², Nami Ogura¹, Tatsuya Suzuki¹, Akiharu Ueki¹, Akio Saito³, Viktor V Zhdankin⁴ (1. Aomori Univ., 2. Tomsk Polytechnic University, 3. Tokyo University of Agriculture and Technology, 4. University of Minneota )

[29P-pm029] Development of the cyclization reaction with alkene and trifluoroacetamide group as radical precursor mediated by samarium(II) diiodide

○Hiroki Iwasaki¹, Saho Ito¹, Yuzuha Iwamoto¹, Hisanori Nambu¹ (1. Kyoto Pharmaceutical Univ.)

[29P-pm030] Alkylidene transfer from 1,3-dipoles to iminoiodanes

○Noriko Okamoto¹, Haruto Ogino¹, Keiji Konishi¹, Takuya Sueda¹ (1. Hiroshima International University)

[29P-pm031S] Development of synthesis for α-amino-β-lactam equivalent using N-Alkynylimide via the Kinugasa reaction

○Chie Nakamo¹, Keiji Konishi¹, Noriko Okamoto¹, Takuya Sueda¹ (1. Hiroshima International University)

[29P-pm032] Regioselective [3+2] Cycloaddition of Ynimides with Azomethine Imines to Generate N,N-Bicyclic 3-Pyrazolidinones

○Risako Hashimoto¹, Keiji Konishi¹, Noriko Okamoto¹, Takuya Sueda¹ (1. Hiroshima International University)

[29P-pm033] Environmentally benign thio-Michael reaction using acidic resin

○Yasunari Monguchi¹, Arisa Kumagai¹, Yuki Yoshida¹, Shuri Yokotake¹, Aika Matsuzono¹, Natsuki Matsumura¹, Kazutaka Koga¹, Sayuri Yokoyama¹ (1. Daiichi University of Pharmacy)

[29P-pm034] A general strategy for nucleophilic fluorination with Et₃N・3HF complex via Halogen exchange

○Satoshi Mizuta¹, Takeshi Ishikawa² (1. Grad. Sch. Biomed. Sci., Nagasaki Univ., 2. Grad. Sch. Sci. Eng., Kagoshima Univ.)

[29P-pm035S] Kharasch addition to α,β-unsaturated oximes

Yuki Honda¹, ○Tomohiro Hitoe¹, Ayaka Yamamoto¹, Yoshimitsu Hashimoto¹, Kosaku Tanaka Ⅲ¹, Nobuyoshi Morita¹, Osamu Tamura¹ (1. Showa Pharm. Univ.)

[29P-pm036S] Catalytic Direct Synthesis of Primary Amides from Carboxylic Acids Using Hexamethyldisilazane as the Nitrogen Source

○Shunsuke Kataoka¹, Takashi Ohshima¹ (1. Grad. Sch. Pharm. Sci., Kyushu Univ.)

[29P-pm037S] Development of One-Pot Transformation of Silyl Ethers to Nitriles

○Suzuka Kubozono¹, Yuka Tanaka¹, Yusuke Kobayashi¹, Takumi Furuta¹, Shohei Hamada¹ (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-pm038] Samarium-catalyzed pinacol coupling using a visible-light-absorbing antenna ligand

○Takahito Kuribara¹, Ayahito Kaneki¹, Yu Matsuda¹, Tetsuhiro Nemoto¹ (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[29P-pm039] Synthesis of azoxybenzene derivatives from nitroarenes via a reductive reaction using a catalytic amount of azastibocine

○yuki murata¹, Seiya Nakashima¹, Tomohiro Fujita¹, Mio Matsumura¹, Shuji Yasuike¹ (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[29P-pm040] Copper-catalyzed three component Se-arylation of selenium powder with pyrazolones and triarylbismuthanes

○Mio Matsumura¹, Ayaka Nakamura¹, Atsuki Yanagida¹, Yuki Murata¹, Shuji Yasuike¹ (1. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[29P-pm041S] Synthesis of novel benzoxazoloisoquinoliniums and optical properties

○Masato Kawakubo¹, Megu Morishita², Yuki Ohno², Yuki Murata², Mio Matsumura², Shuji Yasuike² (1. Grad. Sch. Pharm. Sci., Aichi Gakuin Univ., 2. Sch. Pharm. Sci., Aichi Gakuin Univ.)

[29P-pm042S] Synthesis of triphenylamines bearing a silicon substituent at the ortho position

○Yuria Sato¹, Hikaru Fujita¹, Shiori Kobayashi¹, Munetaka Kunishima^1,2 (1. Faculty of Pharmaceutical Sciences, Institute of Medical, Pharmaceutical, and Health Sciences, Kanazawa University, 2. Faculty of Pharmaceutical Sciences, Kobe Gakuin University)

[29P-pm043] Manganese(III)-catalyzed diastereoselective oxygenative aminoperoxidation

○Daisuke Yamamoto¹, Yuki Narushima¹, Issei Hirano¹, Masayuki Soga¹, Hiromasa Ansai¹, Kazuishi Makino¹ (1. School of Pharmacy, Kitasato Univ.)

[29P-pm044S] Hydrosilylation of Selenoesters and Its Synthetic Application

○Mustapha Kobina Abeka¹, Alex Boateng¹, Yuhei Ohta¹, Masaharu Sugiura¹ (1. Dept. Pharm. Sci., Sojo University)

[29P-pm045S] Development of highly efficient bifunctional asymmetric organocatalyst from conformationally rigid cis-1,2-diamines
~Search for hydrogen bond donor sites~

○Yuki Kurosawa¹, Kento Muneta¹, Satsuki Matsumoto¹, Takuro Yasuyama¹, Hirofumi Matsunaga¹ (1. Fac. Pharm. Sci., Sanyo-Onoda City Univ.)

[29P-pm046S] Development of asymmetric organocatalyst with cis-1,2-diamine framework derived from indane skeleton

○Yuki Yamada¹, Naoki Kawakami¹, Rei Hodumi¹, Takuro Yasuyama¹, Hirofumi Matsunaga¹ (1. Fac. Pharm. Sci., Sanyo-Onoda City Univ.)

[29P-pm047S] Synthesis of β-carboline via oxidative Pictet-Spengler reactions/DBU-mediated aerobic oxidation cascade

○Masakazu Kobayashi¹, Shoko Kikkawa¹, Isao Azumaya¹, Hidemasa Hikawa¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm048S] Au(Ⅲ)-catalyzed dehydrative Bischler-Möhlau type indole synthesis

○Yuuka Kumono¹, Taku Nakayama¹, Shoko Kikkawa¹, Isao Azumaya¹, Hidemasa Hikawa¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm049S] Construction of imidazopyridine skeleton via Pd-catalyzed dehydrogenative oxidation of benzyl alcohol in water

○Nanoka Kobori¹, Masakazu Kobayashi¹, Taku Nakayama¹, Shoko Kikkawa¹, Isao Azumaya¹, Hidemasa Hikawa¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm050S] Dehydrative/decarboxylative coupling of quinoline-4-carboxylic acids with allylic alcohols in water

○En Kenmochi¹, Taku Nakayama¹, Tomokatsu Enda¹, Shoko Kikkawa¹, Isao Azumaya¹, Hidemasa Hikawa¹ (1. Fac. Pharm. Sci. Toho Univ.)

[29P-pm051S] Extension of the Newman-Kwart Rearrangement to Heterocycles

○Yuma Okuda¹, Keita Yamazaki¹, Tetsuhiro Nemoto¹ (1. Grad. Sch. Pharm. Sci., Chiba Univ.)

[29P-pm052S] HFIP accelerates the oxidation of alcohol using TEMPO and PIDA

○Kaori Sakamoto¹, Wakana Oda¹, Yusuke Kobayashi¹, Takumi Furuta¹, Shohei Hamada¹ (1. Fac. Pharm., Kyoto Pharmaceutical University)

[29P-pm053S] Investigation of intermolecular anti-Markownikov Wacker-type reaction

Yasuhiro Nishikawa¹, ○Sayaka Suzuki¹, Momoka Suzuki¹, Sara Kawanishi¹, Kazuma Mizuno¹, Mikako Aoki¹, Osamu Hara¹ (1. Fac. Pharm. , Meijo Univ.)

[29P-pm054S] The development of trivalent bismuth catalyzed oxidative coupling for arenols

Kengo Kasama¹, ○HaoYang Dai¹, Kousuke Umezawa¹, Takayuki Yakura¹ (1. University of Toyama)

[29P-pm055S] Site-selective deuteration of thioacetals using a potassium deuteroxide solution in D₂O

○Hyoga Shimizu¹, Shuji Akai², Yoshinari Sawama^2,3 (1. Sch. Pharm. Sci., Osaka Univ., 2. Grad. Sch. Pharm. Sci., Osaka Univ., 3. Deuterium Science Research Unit, Center for the Promotion of Interdisciplinary Education and Research, Kyoto University)

[29P-pm056S] Palladium-catalyzed construction of B,N-naphthalene scaffold

Yuto Iseya¹, Ryotaro Kume¹, ○Ryo Yanagida², Ozora Sasamoto^1,3, Yoshinori Kondo¹, Masanori Shigeno^1,4 (1. Grad. Sch. Pharm. Sci., Tohoku Univ., 2. Pharm. Sci., Tohoku Univ., 3. RCPD, 4. PRESTO, JST)

[29P-pm057S] Catalyst-Free Aziridination using In Situ Generated Iminoiodanes

○Asaka Kodama¹, Shun Sunagawa¹, Akira Tsubouchi¹, Akio Saito¹ (1. Grad. Sch. Eng., Tokyo Univ. Agric. Tech.)

[29P-pm058] Generation and Cycloaddition of Functionalized Arynes Generated from o-Triazenylarylboronic Acids

○Motoki Ito¹, Haruna Yamazaki¹, Yuta Takishima¹, Aguri Ito¹, Ryuhei Oda¹, Moeka Komiya¹, Kazuhiro Higuchi¹, Shigeo Sugiyama¹ (1. Meiji Pharmaceutical Univ.)

[29P-pm059S] Reactions for the introduction of perfluoroalkyl groups into carbonyl compounds

Tsuyoshi Yamada¹, ○Mana Kumazawa¹, Yutaro Yamada¹, Takashi Ikawa¹, Hironao Sajiki¹ (1. Gifu. Pharm. Univ.)

[29P-pm060S] Synthesis of 1,2-dihydroisoquinoline derivatives by palladium-catalyzed cascade cyclization of allenamides and arylboronic acids

○Ryunosuke Imaji¹, Shinya Shiomi¹, Masahiro Yoshida¹ (1. Faculty of Pharmaceutical Sciences, Tokushima Bunri University)

[29P-pm061S] Development of a new method for constructing benzazetine using dual-wavelength light irradiation

○Kaito Nakajima¹, Masaru Tanioka¹, Yuji Matsuya¹ (1. Faculty of Pharm. Sci., University of Toyama)

[29P-pm062S] Nitrogen-containing heterocycle synthesis utilizing the nucleophilic imino carbon of the hydrazone

○Ayano Ichimonji¹, Miku Nakayama¹, Norihiko Takeda¹, Motohiro Yasui¹, Hiroshi Matsubara², Masafumi Ueda¹ (1. Kobe Pharmaceutical University, 2. Osaka Metropolitan University)

Session information

[29P-pm] Chemical reaction development 1

Authentication